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Tegginamath Gireesh
Articles written in Journal of Chemical Sciences
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Volume 123 Issue 4 July 2011 pp 393-401
An efficient synthesis, X-ray and spectral characterization of biphenyl derivatives
Ravindra R Kamble Dharesh B Biradar Gangadhar Y Meti Tasneem Taj Tegginamath Gireesh Imthiyaz Ahmed M Khazi Sundar T Vaidyanathan Raju Mohandoss Balasubramanian Sridhar Viraraghav Parthasarathi
Derivatives of 1,3-thiazolidin-2,4-dione appended to biphenyl ring viz., 7-9, 16-18 were prepared. The newly synthesized compounds were confirmed by IR, NMR (1H and 13C) MS and elemental analyses. Single crystal X-ray diffraction study was carried out for one of the final compounds 9.
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Volume 123 Issue 5 September 2011 pp 657-666
An expeditious green synthesis of Schiff bases and azetidinones derivatised with 1,2,4-triazoles
Tasneem Taj Ravindra R Kamble Tegginamath Gireesh Bharathi V Badami
An efficient green approach to the synthesis of Schiff bases (
11-21 ) of 1-amino-2-aryl-3-oxo-1,2,4-triazoles (1-3 ) have been reported under Mg(ClO4)2 as catalyst followed by the reaction with chloroacetyl chloride in solvent-free conditions to yield the azetidinones (22-32 ) with excellent yields. The synthesized compounds were evaluated for the extent of penetration into biological membranes ($clogP$), drug-likeliness and finally drug score was calculated and also screened for antitubercular and antimicrobial activities.
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Journal of Chemical Sciences
Volume 135, 2023
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